Email this article 
Hide
Show all
OPEN ACCESS | 
PEER-REVIEWED |
RESEARCH ARTICLE
|
DOWNLOAD PDF
|
VIEW FULL-TEXT PDF
| TOTAL VIEWS
NaOH/PEG-400: An eloquent system for the synthesis of new thienyl benzo[b]1,4-diazepines
Gajanan Gopinath Mandawad (1)
, Baseer Mubeen Shaikh (2) , Santosh Subhash Chobe (3) , Shankaraiah Guruvaiah Konda (4,*) (1) Department of Chemistry, Maharashtra Udayagiri College, Udgir-413517, Maharashtra, India
(2) Department of Chemistry, Sir Sayyed College, Aurangabad-431001, Maharashtra, India
(3) Organic Research Laboratory, Loknete Vyankatrao Hirey College, Nashik-422003, Maharashtra, India
(4) Department of Chemistry, Karamsibhai Jethabhai Somaiya College, Kopargaon-423601, Maharashtra, India
(*) Corresponding Author
Received: 19 Jul 2020 | Revised: 05 Sep 2020 | Accepted: 14 Sep 2020 | Published: 31 Dec 2020 | Issue Date: December 2020
Abstract
A simple and eloquent procedure for the synthesis of a new series of thienyl benzo[b]1,4-diazepines is reported. They were synthesized by the condensation of o-phenylenediamine (o-PDA) with distinct hetero chalcones using NaOH in polyethylene glycol (PEG-400) as green and alternative reaction solvent. The significances of this present method are shorter reaction time, easy work-up, high yields, and mild reaction conditions. Furthermore, this method is environment friendly and without use of an expensive catalyst. The all newly synthesized compounds are characterized by the spectroscopic methods.
Announcements
One of our sponsors will cover the article processing fee for all submissions made between May 17, 2023 and June 16, 2023 (Voucher code: SPONSOR2023).
Editor-in-Chief
European Journal of Chemistry
Keywords
Full Text:
PDF
DOI: 10.5155/eurjchem.11.4.276-279.2009
Links for Article
| | | | | | |
| | | | | | |
| | | |
Related Articles
Article Metrics
This Abstract was viewed 889 times |
PDF Article downloaded 416 times
Citations
[1]. Sunita Teli, Pankaj Teli, Shivani Soni, Nusrat Sahiba, Shikha Agarwal
Synthetic aspects of 1,4- and 1,5-benzodiazepines using o-phenylenediamine: a study of past quinquennial
RSC Advances 13(6), 3694, 2023
DOI: 10.1039/D2RA06045K
[2]. Shankaraiah G. Konda, Santosh S. Chobe, Amit Kumar N. Gosar, Baliram S. Hote,, Gajanan G. Mandawad
Polyethylene Glycol-400 Prompted an Efficient Synthesis of Thienyl Pyrazolo[ 1,5‐a] Pyrimidines as Microbial Inhibitors
Current Organic Synthesis 19(6), 693, 2022
DOI: 10.2174/1570179419666220304160938
References
[1]. Mallinath, M. L. Der Pharma Chem. 2011, 3(2), 273-276.
[2]. Konda, S. G.; Shaikh, B. M.; Chavan, S. A.; Dawane, B. S. Chinese Chem. Lett. 2011, 22, 65-68.
https://doi.org/10.1016/j.cclet.2010.09.012
[3]. Naraboli, B. S.; Biradar, J. S. Int. J. Pharm. Pharm. Sci. 2017, 9(8), 128-138.
https://doi.org/10.22159/ijpps.2017v9i8.19725
[4]. Sandra, C. M.; Eduardo, C. C.; Simon, H. O.; Teresa, R. A.; Antonio, N. C.; Lijanova, I. V. Med. Chem. 2012, 12(6), 611-618.
https://doi.org/10.2174/187152012800617713
[5]. Henderson, E. A.; Alber, D. G.; Baxter, R. C.; Bithell, S. K.; Budworth, J.; Carter, M. C. J. Med. Chem. 2007, 50(7), 1685-1692.
https://doi.org/10.1021/jm060747l
[6]. Griffin, C. E.; Kaye, A. M.; Bueno, F. R.; Kaye, A. D. Ochsner. J. 2013, 13(2), 214-223.
[7]. Thakuria, H.; Pramanik, A.; Borah, B. M.; Das, G. Tetrahedron Lett. 2006, 47, 3135-3138.
https://doi.org/10.1016/j.tetlet.2006.02.137
[8]. Reddy, K. V. V.; Rao, P. S.; Ashok, D. Synth. Commun. 2000, 30, 1825-1836.
[9]. Gupta, R.; Kumar, M.; Gupta, V. Heterocyclic Chemistry of Five Membered Heterocycles, New York, 1999, 2. 416-426.
https://doi.org/10.1007/978-3-662-07757-3
[10]. Herbert, J. A. L.; Suschitzky, H. J. Chem. Soc., Perkin Trans. 1974, 1, 2657-2661.
https://doi.org/10.1039/p19740002657
[11]. Morales, H. R.; Bulbarela, A. Heterocycles 1986, 24, 135-139.
https://doi.org/10.3987/R-1986-01-0135
[12]. Jung, D. I.; Choi, T. W.; Kim, Y. Y.; Kim, I. S.; Park, Y. M.; Lee, Y. G.; Jung, D. H. Synth. Commun. 1999, 29, 1941-1951.
[13]. Yadav, J. S.; Reddy, B. V. S.; Eshwaraian, B.; Anuradha, K. Green Chem. 2002, 4, 592-594.
https://doi.org/10.1039/B206558B
[14]. Curini, M.; Epifano, F.; Marcotullio, M. C.; Rosati, O. Tetrahedron Lett. 2001, 42, 3193-3195.
https://doi.org/10.1016/S0040-4039(01)00413-0
[15]. Balakrishna, M. S.; Kaboundin, B. Tetrahedron Lett. 2001, 42, 1127-1129.
https://doi.org/10.1016/S0040-4039(00)02168-7
[16]. Pozarentzi, M.; Stephanidou, S. J. Tetrahedron Lett. 2002, 43, 1755-1758.
https://doi.org/10.1016/S0040-4039(02)00115-6
[17]. Ma, Y.; Zhang, Y. Synth. Commun. 2002, 32, 163-166.
[18]. Jarikote, D. V.; Siddique, S. A.; Rajagopal, R.; Daniel, T.; Lahoti, R. J.; Srinivasan, K. V. Tetrahedron Lett. 2003, 44, 1835-1838.
https://doi.org/10.1016/S0040-4039(03)00096-0
[19]. Kodomari, M.; Noguchi, T.; Aoyama, T. Synth. Commun. 2004, 34, 1783-1790.
https://doi.org/10.1081/SCC-120034159
[20]. Sabitha, G. S.; Reddy, K. K.; Reddy, K. B.; Reddy, N. M.; Yadav, J. S. Adv. Synth. Catal. 2004, 346, 921-923.
https://doi.org/10.1002/adsc.200303196
[21]. Reddy, B. M.; Sreekanth, P. M.; Reddy, V. R. J. Mol. Cat A 2005, 225, 71-78.
https://doi.org/10.1016/j.molcata.2004.09.003
[22]. Kaboudin, B.; Navaee, K. Heterocycles 2001, 55(8), 1443-1446.
https://doi.org/10.3987/COM-01-9253
[23]. Yadav, J. S.; Reddy, B. V. S.; Praveenkumar, S.; Nagaiah, K.; Lingaiah, N.; Saiprasad, P. S. Synthesis 2004, 6, 901-904.
https://doi.org/10.1055/s-2004-816013
[24]. Chari, M. A.; Syamasundar, K. Cat. Commun. 2005, 6(1), 67-70.
https://doi.org/10.1016/j.catcom.2004.10.009
[25]. Hegedus, A.; Hell, Z.; Potor, A. Cat. Lett. 2005, 105, 229-232.
https://doi.org/10.1007/s10562-005-8695-4
[26]. Chen, J.; Spear, S. K.; Huddieston, J. G.; Rogers, R. D. Green Chem. 2005, 7, 64-82.
https://doi.org/10.1039/b413546f
[27]. Heldebrant, D.; Jessop, P. G. J. Am. Chem. Soc. 2003, 125, 5600-5601.
https://doi.org/10.1021/ja029131l
[28]. Chandrasekhar, S.; Narsihmulu, Ch.; Sultana, S. S.; Reddy, N. R. K. Org. Lett. 2002, 4, 4383-4399.
https://doi.org/10.1021/ol0266976
[29]. Jiang, R.; Kuang, Y. Q.; Sun, X. L.; Zhang, S. Y. Tetrahedron Asym. 2004, 15, 743-746.
https://doi.org/10.1016/j.tetasy.2004.01.011
[30]. Namboodiri, V. V.; Varma, R. S. Green Chem. 2001, 3, 146-148.
https://doi.org/10.1039/b102337n
[31]. Suryakiran, N.; Ramesh, D.; Venkateswarulu, Y. Green Chem. Lett. 2007, 1, 73-78.
https://doi.org/10.1080/17518250701771909
[32]. Kamal, A.; Reddy, D. R.; Rajendar, S. Tetrahedron Lett. 2005, 46, 7951-7953.
https://doi.org/10.1016/j.tetlet.2005.09.082
[33]. Kamble, V. T.; Dawane, B. S.; Chavan, S. A.; Bhosale, R. B. Aust. J. Chem. 2007, 60, 302-304.
https://doi.org/10.1071/CH06377
[34]. Das, B.; Krishnaiah, M.; Balasybramanyam, P.; Veeranjaneyulu, B.; Nanda, K. D. Tetrahedron Lett. 2008, 49, 2225-2227.
https://doi.org/10.1016/j.tetlet.2008.02.050
[35]. Konda, S. G.; Humne, V. T.; Lokhande, P. D. Green Chem. 2011, 13, 2354-2358.
https://doi.org/10.1039/c1gc15153c
[36]. Dawane, B. S.; Konda, S. G.; Bhosale, R. B.; Shaikh, B. M. Acta. Pharm. 2009, 59, 473-482.
https://doi.org/10.2478/v10007-009-0034-7
[37]. Dawane, B. S.; Konda, S. G.; Mandawad, G. G.; Shaikh, B. M. Eur. J. Med. Chem. 2010, 45, 387-392.
[38]. Konda, S. G. Eur. J. Chem. 2014, 5(4), 676-680.
https://doi.org/10.5155/eurjchem.5.4.676-680.1110
[39]. Konda, S. G. J. Adv. Chem. Sci. 2016, 2(3), 363-365.
[40]. Mandawad, G. G.; Chobe, S. S.; Yemul, O. S.; Dawane, B. S. J. Pharm Res. 2011, 4(10), 3360-3363.
How to cite
The other citation formats (EndNote | Reference Manager | ProCite | BibTeX | RefWorks) for this article can be found online at: How to cite item
DOI Link: https://doi.org/10.5155/eurjchem.11.4.276-279.2009
| 
| 
| 
| 
| 
| 
| 
| 
| 
| 
| 
| 
| 
| 
| 
Save to Zotero
Save to Mendeley
European Journal of Chemistry 2020, 11(4), 276-279 | doi: https://doi.org/10.5155/eurjchem.11.4.276-279.2009 | Get rights and content
Refbacks
- There are currently no refbacks.
Copyright (c) 2020 Authors
This work is published and licensed by Atlanta Publishing House LLC, Atlanta, GA, USA. The full terms of this license are available at http://www.eurjchem.com/index.php/eurjchem/pages/view/terms and incorporate the Creative Commons Attribution-Non Commercial (CC BY NC) (International, v4.0) License (http://creativecommons.org/licenses/by-nc/4.0). By accessing the work, you hereby accept the Terms. This is an open access article distributed under the terms and conditions of the CC BY NC License, which permits unrestricted non-commercial use, distribution, and reproduction in any medium, provided the original work is properly cited without any further permission from Atlanta Publishing House LLC (European Journal of Chemistry). No use, distribution or reproduction is permitted which does not comply with these terms. Permissions for commercial use of this work beyond the scope of the License (http://www.eurjchem.com/index.php/eurjchem/pages/view/terms) are administered by Atlanta Publishing House LLC (European Journal of Chemistry).
© Copyright 2010 - 2023 • Atlanta Publishing House LLC • All Right Reserved.
The opinions expressed in all articles published in European Journal of Chemistry are those of the specific author(s), and do not necessarily reflect the views of Atlanta Publishing House LLC, or European Journal of Chemistry, or any of its employees.
Copyright 2010-2023 Atlanta Publishing House LLC. All rights reserved. This site is owned and operated by Atlanta Publishing House LLC whose registered office is 2850 Smith Ridge Trce Peachtree Cor GA 30071-2636, USA. Registered in USA.