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Synthesis and characterization of diaza analogues of podophyllotoxin
Yeriyur Basavaiah Basavaraju (1,*)
, Basavaiah Umesha (2) (1) Department of Studies in Chemistry, University of Mysore, Manasagangotri, Mysore-570006, Karnataka, India
(2) Department of Studies in Chemistry, University of Mysore, Manasagangotri, Mysore-570006, Karnataka, India
(*) Corresponding Author
Received: 23 Mar 2013 | Accepted: 07 May 2013 | Published: 30 Sep 2013 | Issue Date: September 2013
Abstract
In an attempt to synthesize the novel diaza analogues of podophyllotoxin (7a-d) in five step reactions. The synthesis of title compounds has been achieved from tetralones, which were formylated with ethylformate; prepared via cyclization with hydrazine hydrate. Furthermore, these newly synthesized compounds were characterized by spectral and elemental analysis data.
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European Journal of Chemistry
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DOI: 10.5155/eurjchem.4.3.235-239.782
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Funding information
Indian Institute of Technology, Bombay, India
Citations
[1]. Basavaiah Umesha, Yeriyur Basavaiah Basavaraju, Manpreet Kaur, Hemmige S. Yathirajan, Jerry P. Jasinski
1-(3,4-Dimethoxyphenyl)-3-phenylprop-2-en-1-one
Acta Crystallographica Section E Structure Reports Online 70(3), o368, 2014
DOI: 10.1107/S160053681400378X
[2]. Krishna Mudeenahally Hucchegowda, Basavaraju Yeriyur Basavaiah, Umesha Basavaiah, Shivakumar Santhekasalagere Basavaiah
Synthesis and study of antimicrobial activity of new tetralone esters
European Journal of Chemistry 5(4), 584, 2014
DOI: 10.5155/eurjchem.5.4.584-587.1093
[3]. Kanakapura Narayanaramakrishna Padmavath, Yeriyuru Basavaiah Basavaraju, Basavaiah Umesha
Synthesis and characterization of tetralones as intermediates for podophyllotoxin analogues
European Journal of Chemistry 7(2), 192, 2016
DOI: 10.5155/eurjchem.7.2.192-194.1389
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DOI Link: https://doi.org/10.5155/eurjchem.4.3.235-239.782
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European Journal of Chemistry 2013, 4(3), 235-239 | doi: https://doi.org/10.5155/eurjchem.4.3.235-239.782 | Get rights and content
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