European Journal of Chemistry

Activated bentonite promoted Friedländer condensation reactions: Synthesis of thieno[2,3-b]quinolinones and tacrines analogues derivatives



Main Article Content

Khaireddine Mohamed Dridi
Ridha Ben Said
Youssef Arfaoui
Abdullah Sulaiman Al-Ayed

Abstract

Some new aminothieno[2,3-b]quinolinones and tacrine analogues derivatives were synthesized in high yield with acid activated bentonite as a catalyst via the Friedländer condensation reactions between 2-aminothiophene-3-carbonitrile and ketones. The structure elucidation of compounds was done by FT-IR, NMR spectroscopy and microanalytical elemental data.

4_3_216_219

icon graph This Abstract was viewed 1700 times | icon graph Article PDF downloaded 788 times

How to Cite
(1)
Dridi, K. M.; Said, R. B.; Arfaoui, Y.; Al-Ayed, A. S. Activated Bentonite Promoted Friedländer Condensation Reactions: Synthesis of thieno[2,3-b]quinolinones and Tacrines Analogues Derivatives. Eur. J. Chem. 2013, 4, 216-219.

Article Details

Share
Crossref - Scopus - Google - European PMC
References

[1]. Summers, W. K.; Majovsky, L. V.; Marsh, G. M.; Tachiki, K.; Kling, A. N. Engl. J. Med. 1986, 315, 1241-1287
http://dx.doi.org/10.1056/NEJM198611133152001
PMid:2430180

[2]. Sahakian, B. J.; Owen, A. M.; Morant, N. J.; Eagger, S. A.; Boddington, S.; Crayton, L.; Crockford, H. A.; Crooks, M.; Hill, K.; Levy, R. Psychopharmacology 1993, 110, 395-401.
http://dx.doi.org/10.1007/BF02244644

[3]. Drukarch, B.; Kits, K. S.; Van der Meer, E. G.; Lodder, J. C.; Stoof, J. C. Eur. J. Pharmacol. 1987, 141, 153-157.
http://dx.doi.org/10.1016/0014-2999(87)90424-9

[4]. Augry, F.; Darch, A.; De Routou, J.; Guelfi, M. C.; Forette, F. J. Pharm. Clin. 1997, 16, 183-201.

[5]. Dridi, K.; El Efrit, M. L.; Zantour, H. J. Soc. Chim. Tunisie 1999, 5, 387-392.

[6]. Dridi, K.; El Efrit, M. L.; Zantour, H. J. Soc. Chim. Tunisie 2001, 4, 957-963.

[7]. Gutschow, M.; Kuerschner, L.; Neumann, U.; Peitsch, M.; Loser, R.; Koglin, N.; Eger, K. J. Med. Chem. 1999, 42, 5437-5447.
http://dx.doi.org/10.1021/jm991108w

[8]. Fugita, M.; Seki, T.; Ikeda, N. Bioorg. Med. Chem. Lett. 2002, 12, 1897-1900.
http://dx.doi.org/10.1016/S0960-894X(02)00332-3

[9]. Harza, K.; Saravanan, J.; Mohan, S. Asian J. Chem. 2007, 19, 3541-3544.

[10]. Narlawar, R.; Lane, J. R.; Doddareddy, M.; Lin, J.; Brussee, J.; Ijzerman, A. P. J. Med. Chem. 2010, 53, 3028-3037.
http://dx.doi.org/10.1021/jm901252a
PMid:20345101

[11]. Marco-Contelles, J.; Perez-Mayoral, E.; Samadi, A.; Carreiras, M. C.; Soriano, E. Chem. Rev. 2009, 109, 2652-2671.
http://dx.doi.org/10.1021/cr800482c
PMid:19361199

[12]. Laszlo, P.; Mathy, A. Hel. Chim. Acta 1987, 70, 577-586.
http://dx.doi.org/10.1002/hlca.19870700310

[13]. Choudary, B. M.; Kantam, M. L.; Rao, K. K.; Santhi, P. L. Appl. Catal. A. Gen. 1997, 149, 257-264.
http://dx.doi.org/10.1016/S0926-860X(96)00310-9

[14]. Yoo, J. W.; Lee, C. W.; Jeong, H. C.; Park, Y. K.; Park, S. E. Catal. Today 2000, 60, 255-261.
http://dx.doi.org/10.1016/S0920-5861(00)00342-4

[15]. Inui, K.; Kurabayashi, T.; Sato, S.; Ichikawa, N. J. Mol. Catal. A 2006, 216, 147-155.
http://dx.doi.org/10.1016/j.molcata.2004.02.017

[16]. Gewald, K.; Schinke, E.; Bohcher, H. Chem. Ber. 1966, 99, 94-100.
http://dx.doi.org/10.1002/cber.19660990116

[17]. Eller, G. A.; Wolfgang, H. Molecules 2006, 11, 371-376.
http://dx.doi.org/10.3390/11050371
PMid:17962769

Supporting Agencies

The Deanship of Scientific Research at Qassim University, Project No, 1799, Qassim University, AlRass, 53, Kingdom of Saudi Arabia
Most read articles by the same author(s)
TrendMD

Dimensions - Altmetric - scite_ - PlumX

Downloads and views

Downloads

Download data is not yet available.

Metrics

Metrics Loading ...
License Terms

License Terms

by-nc

Copyright © 2024 by Authors. This work is published and licensed by Atlanta Publishing House LLC, Atlanta, GA, USA. The full terms of this license are available at https://www.eurjchem.com/index.php/eurjchem/terms and incorporate the Creative Commons Attribution-Non Commercial (CC BY NC) (International, v4.0) License (http://creativecommons.org/licenses/by-nc/4.0). By accessing the work, you hereby accept the Terms. This is an open access article distributed under the terms and conditions of the CC BY NC License, which permits unrestricted non-commercial use, distribution, and reproduction in any medium, provided the original work is properly cited without any further permission from Atlanta Publishing House LLC (European Journal of Chemistry). No use, distribution, or reproduction is permitted which does not comply with these terms. Permissions for commercial use of this work beyond the scope of the License (https://www.eurjchem.com/index.php/eurjchem/terms) are administered by Atlanta Publishing House LLC (European Journal of Chemistry).