European Journal of Chemistry

Activated bentonite promoted Friedländer condensation reactions: Synthesis of thieno[2,3-b]quinolinones and tacrines analogues derivatives

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Published: Sep 30, 2013
DOI: https://doi.org/10.5155/eurjchem.4.3.216-219.788
Keywords:
Ketones, Bentonite, Tacrine analogues, Friedlander reaction, 2-Aminothiophene-3-carbonitrile, 4-Aminothieno[2, 3-b]quinolinones
Section
Research Article
Issue
Vol. 4 No. 3 (2013): September 2013
Dates
Received 2013-04-01
Accepted 2013-05-08
Published 2013-09-30


Main Article Content

Khaireddine Mohamed Dridi
Department of Chemistry, College of Sciences and Arts, Qassim University, Al-Rass, 53, Kingdom of Saudi Arabia
Ridha Ben Said
Unité Physico-Chimie des Matériaux Condensés, Département de Chimie, Faculté des Sciences, Université Tunis El Manar, El Manar II, Tunis 1060, Tunisia
Youssef Arfaoui
Unité Physico-Chimie des Matériaux Condensés, Département de Chimie, Faculté des Sciences, Université Tunis El Manar, El Manar II, Tunis 1060, Tunisia
Abdullah Sulaiman Al-Ayed
Department of Chemistry, College of Sciences and Arts, Qassim University, Al-Rass, 53, Kingdom of Saudi Arabia

Abstract

Some new aminothieno[2,3-b]quinolinones and tacrine analogues derivatives were synthesized in high yield with acid activated bentonite as a catalyst via the Friedländer condensation reactions between 2-aminothiophene-3-carbonitrile and ketones. The structure elucidation of compounds was done by FT-IR, NMR spectroscopy and microanalytical elemental data.

4_3_216_219

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Dridi, K. M.; Said, R. B.; Arfaoui, Y.; Al-Ayed, A. S. Activated Bentonite Promoted Friedländer Condensation Reactions: Synthesis of thieno[2,3-b]quinolinones and Tacrines Analogues Derivatives. Eur. J. Chem. 2013, 4, 216-219.

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Supporting Agencies

The Deanship of Scientific Research at Qassim University, Project No, 1799, Qassim University, AlRass, 53, Kingdom of Saudi Arabia
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