European Journal of Chemistry 2013, 4(2), 98-101 | doi: https://doi.org/10.5155/eurjchem.4.2.98-101.714 | Get rights and content






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Synthesis and antimicrobial activity of some novel 2-azetidinones and 4-thiazolidinones derivatives


Shivaji Chavan (1) , Sainath Zangade (2) , Archana Vibhute (3) , Yeshwant Vibhute (4,*)

(1) Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
(2) Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
(3) Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
(4) Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
(*) Corresponding Author

Received: 02 Dec 2012 | Revised: 08 Jan 2013 | Accepted: 08 Jan 2013 | Published: 30 Jun 2013 | Issue Date: June 2013

Abstract


Several 2-azetidinones 2a-e and 4-thiazolidinones 3a-e have been synthesized from halo-substituted Schiff bases using conventional as well as microwave technique. The newly synthesized compounds were established on the basis of spectroscopic technique. Further, all compounds screened for antimicrobial activity against Bacillus subtilis, Escherichia coli, Aspergillus niger and Aspergillus flavus. Most of the titled compounds show potent activity.

4_2_98_101

Keywords


Synthesis; 2-Azetidinones; 4-Thiazolidinones; Microwave technique; Antimicrobial activity; Halosubstituted Schiff bases

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DOI: 10.5155/eurjchem.4.2.98-101.714

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Funding information


University Grant Commission (No. 38‐267/2009), New Delhi, India

Citations

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[1]. Javeed Ahmad War, Santosh Kumar Srivastava, Savitri Devi Srivastava
Design, synthesis and molecular docking studies of some morpholine linked thiazolidinone hybrid molecules
European Journal of Chemistry  7(3), 271, 2016
DOI: 10.5155/eurjchem.7.3.271-279.1427
/


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How to cite


Chavan, S.; Zangade, S.; Vibhute, A.; Vibhute, Y. Eur. J. Chem. 2013, 4(2), 98-101. doi:10.5155/eurjchem.4.2.98-101.714
Chavan, S.; Zangade, S.; Vibhute, A.; Vibhute, Y. Synthesis and antimicrobial activity of some novel 2-azetidinones and 4-thiazolidinones derivatives. Eur. J. Chem. 2013, 4(2), 98-101. doi:10.5155/eurjchem.4.2.98-101.714
Chavan, S., Zangade, S., Vibhute, A., & Vibhute, Y. (2013). Synthesis and antimicrobial activity of some novel 2-azetidinones and 4-thiazolidinones derivatives. European Journal of Chemistry, 4(2), 98-101. doi:10.5155/eurjchem.4.2.98-101.714
Chavan, Shivaji, Sainath Zangade, Archana Vibhute, & Yeshwant Vibhute. "Synthesis and antimicrobial activity of some novel 2-azetidinones and 4-thiazolidinones derivatives." European Journal of Chemistry [Online], 4.2 (2013): 98-101. Web. 3 Jun. 2020
Chavan, Shivaji, Zangade, Sainath, Vibhute, Archana, AND Vibhute, Yeshwant. "Synthesis and antimicrobial activity of some novel 2-azetidinones and 4-thiazolidinones derivatives" European Journal of Chemistry [Online], Volume 4 Number 2 (30 June 2013)

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DOI Link: https://doi.org/10.5155/eurjchem.4.2.98-101.714

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