European Journal of Chemistry

Synthesis and antimicrobial activity of some novel 2-azetidinones and 4-thiazolidinones derivatives

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Published: Jun 30, 2013
DOI: https://doi.org/10.5155/eurjchem.4.2.98-101.714
Keywords:
Synthesis, 2-Azetidinones, 4-Thiazolidinones, Microwave technique, Antimicrobial activity, Halosubstituted Schiff bases
Section
Research Article
Issue
Vol. 4 No. 2 (2013): June 2013
Dates
Received 2012-12-02
Accepted 2013-01-08
Published 2013-06-30


Main Article Content

Shivaji Chavan
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
Sainath Zangade
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
Archana Vibhute
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
Yeshwant Vibhute
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India

Abstract

Several 2-azetidinones 2a-e and 4-thiazolidinones 3a-e have been synthesized from halo-substituted Schiff bases using conventional as well as microwave technique. The newly synthesized compounds were established on the basis of spectroscopic technique. Further, all compounds screened for antimicrobial activity against Bacillus subtilis, Escherichia coli, Aspergillus niger and Aspergillus flavus. Most of the titled compounds show potent activity.

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How to Cite
(1)
Chavan, S.; Zangade, S.; Vibhute, A.; Vibhute, Y. Synthesis and Antimicrobial Activity of Some Novel 2-Azetidinones and 4-Thiazolidinones Derivatives. Eur. J. Chem. 2013, 4, 98-101.

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References

[1]. Dave, T. K.; Purohit, D. H.; Akbari, J. D.; Joshi, S. H. Indian J. Chem. 2007, 46B, 352-356.

[2]. Patel, R. B.; Desai, P. S.; Desai, K. R.; Chikhalia, K. H. Indian J. Chem. 2006, 45B, 773-778.

[3]. Vijay, K. M. M. J.; Nagaraja, T. S.; Shameer, H.; Jayachandran, E.; Sreenivasa, G. M. J. Pharm. Sci. Res. 2009, 1, 83-92.

[4]. Udupi, R. H.; Kasinath, N.; Bhat, A. R. Indian J. Heterocycl. Chem. 1998, 17, 221-224.

[5]. Singh, G. S.; Mbukwa, E.; Pheko, T. Arkivoc 2007, 9, 80-90.

[6]. Chavan, A. A.; Pai, N. R. Molecules 2007, 12, 2467-2477.
http://dx.doi.org/10.3390/12112467
PMid:18065951

[7]. Havaldar, F. H.; Mishra, S. J. Indian J. Heterocycl. Chem. 2004, 13, 197-200.

[8]. Patel, K. H.; Metha, A. G. E-J. Chem. 2006, 3, 267-273.

[9]. Trautman, H. D.; Longe, L. M. J. Am. Chem. Soc. 1948, 70, 3436-3439.
http://dx.doi.org/10.1021/ja01190a064

[10]. Surray, A. R. J. Am. Chem. Soc. 1949, 71, 3354-3356.
http://dx.doi.org/10.1021/ja01178a023

[11]. French, G. Chem. Abstr. 1966, 65, 4439-4445.

[12]. Doran, W. J.; Sholen, H. A. J. Org. Chem. 1938, 3, 193-197.
http://dx.doi.org/10.1021/jo01220a001

[13]. Kuçukguzel, G.; Kocatepe, A.; De Clercq, E.; Sahin, F.; Gulluce, M. Eur. J. Med. Chem. 2006, 41, 353-359.
http://dx.doi.org/10.1016/j.ejmech.2005.11.005
PMid:16414150

[14]. Yadav, R.; Srivastav, S. D.; Srivastav, S. K. Indian J. Chem. 2005, 44B, 1262-1266.

[15]. Oza, H.; Joshi, D. Parekh, H. Indian J. Chem. 1998, 37B, 822-824.

[16]. Saundane, A. R.; Yarlakatti, M.; Walmik, P.; Katkar, V. J. Chem. Sci. 2012, 124, 469-481.
http://dx.doi.org/10.1007/s12039-011-0180-6

[17]. Patel, R. B.; Desai, P. S.; Desai, K. R.; Chikhalia, K. H. Indian J. Chem. B 2006, 45, 773-778.

[18]. Solankee, A. N.; Patel, K. P.; Patel, R. B. Pelagia Res. Lib. 2012, 3, 117-122.

[19]. Bouzroura, S.; Bentarzi, Y.; Kaoua, R.; Nedjar-koli, B.; Poulain-Martini, S.; Dunach, E. Org. Commun. 2010, 3, 8-14.

[20]. Zangade, S. B.; Mokle, S. S.; Shinde, A. T.; Vibhute, Y. B. Green Chem. Lett. Rev. 2013, 6, 123-127.
http://dx.doi.org/10.1080/17518253.2012.713123

[21]. Zangade, S.; Shinde, A.; Patil, A.; Vibhute, Y. Eur. J. Chem. 2012, 3, 208-210.
http://dx.doi.org/10.5155/eurjchem.3.2.208-210.581

[22]. Karamunge, K. G.; Sayed, M. A.; Vibhute, A. Y.; Vibhute, Y. B. J. Indian. Chem. Soc. 2011, 88, 443-446.

[23]. Zangade, S.; Mokle, S.; Chavan, S.; Vibhute, Y. Orbital: Electronic J. Chem. 2011, 3, 144-149.

[24]. Zangade, S. B.; Shinde, A. T.; Vibhute, A. Y.; Vibhute, Y. B. Pak. J. Chem. 2012, 2(1), 18-23.

[25]. Chavan, S. B.; Zangade, S. B.; Vibhute, A. Y. Vibhute, Y. B. Research J. Pharm. Bio. Chem. Sci. 2012, 3, 262-269.

[26]. Bouzroura, S.; Bentarzi, Y.; Kaoua, R.; Nedjar-Kolli, B.; Poulain-Martini, S.; Dunach, E. Org. Commun. 2010, 3(1), 8-14.

[27]. Pawar, R. P.; Andurkar, N. M.; Vibhute, Y. B. J. Indian. Chem. Soc. 1999, 76, 271-272.

[28]. Shinde, A. T.; Zangade, S. B.; Chavan, S. B.; Vibhute, A. Y.; Nalwar, Y. S.; Vibhute, Y. B. Synth. Commun. 2010, 40, 3506-3513.
http://dx.doi.org/10.1080/00397910903457332

[29]. Varma, S. Green Chem. 1999, 1, 43-55.
http://dx.doi.org/10.1039/a808223e

[30]. Borah, R.; Kalita, D. J.; Sarma J. C. Indian J. Chem. B 2002, 41, 1032-1038.

Supporting Agencies

University Grant Commission (No. 38‐267/2009), New Delhi, India
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